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GENE - CHEMICAL INTERACTIONS REPORT

RGD ID: 2520
Species: Rattus norvegicus
RGD Object: Gene
Symbol: Drd2
Name: dopamine receptor D2
Acc ID: CHEBI:8207
Term: (+)-pilocarpine
Definition: The (+)-enantiomer of pilocarpine.
Chemical ID: MESH:D010862
Note: Use of the qualifier "multiple interactions" designates that the annotated interaction is comprised of a complex set of reactions and/or regulatory events, possibly involving additional chemicals and/or gene products.
Object SymbolQualifierEvidenceWithReferenceSourceNotesOriginal Reference(s)
Drd2decreases activityEXP 6480464CTDPilocarpine results in decreased activity of DRD2 proteinPMID:15876489
Drd2decreases expressionEXP 6480464CTDPilocarpine results in decreased expression of DRD2 proteinPMID:15876489
Drd2decreases response to substanceEXP 6480464CTDDRD2 protein results in decreased susceptibility to PilocarpinePMID:1365435
Drd2multiple interactionsEXP 6480464CTD[[Remoxipride results in decreased activity of DRD2 protein] co-treated with [N-(2-(4-(2-methoxyphenyl)-1-piperazinyl)ethyl)-N-(2-pyridinyl)cyclohexanecarboxamide results in decreased activity of HTR1A protein]] results in increased susceptibility to Pilocarpine; [Remoxipride results in decreased activity of DRD2 protein] inhibits the reaction [Dopamine results in decreased susceptibility to Pilocarpine]; Pilocarpine inhibits the reaction [Spiperone binds to DRD2 protein]; Pilocarpine promotes the reaction [Spiperone binds to DRD2 protein]PMID:14559291 PMID:15140183 PMID:16137708
Drd2decreases response to substanceISODrd2 (Mus musculus)6480464CTDDRD2 protein results in decreased susceptibility to PilocarpinePMID:11860278
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