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GENE - CHEMICAL INTERACTIONS REPORT

RGD ID: 2332
Species: Rattus norvegicus
RGD Object: Gene
Symbol: Cftr
Name: CF transmembrane conductance regulator
Acc ID: CHEBI:34756
Term: fenamic acid
Definition: An aminobenzoic acid that is the N-phenyl derivative of anthranilic acid. It acts as a parent skeleton for the synthesis of several non-steroidal anti-inflammatory drugs.
Chemical ID: MESH:C001209
Note: Use of the qualifier "multiple interactions" designates that the annotated interaction is comprised of a complex set of reactions and/or regulatory events, possibly involving additional chemicals and/or gene products.
Object SymbolQualifierEvidenceWithReferenceSourceNotesOriginal Reference(s)
Cftrdecreases activityEXP 6480464CTDfenamic acid results in decreased activity of CFTR proteinPMID:15020588
Cftrdecreases activityISOCftr (Mus musculus)6480464CTDfenamic acid results in decreased activity of CFTR proteinPMID:15986093
Cftrdecreases activityISOCFTR (Homo sapiens)6480464CTDfenamic acid results in decreased activity of CFTR proteinPMID:14502435 PMID:14668136 PMID:15277574 PMID:15857825 PMID:15921678
Cftrmultiple interactionsISOCFTR (Homo sapiens)6480464CTDfenamic acid inhibits the reaction [[[Colforsin co-treated with Genistein] results in increased activity of CFTR protein] which results in increased transport of Iodides]; fenamic acid inhibits the reaction [Colforsin results in increased activity of CFTR protein]PMID:16038730 PMID:18230692
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