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GENE - CHEMICAL INTERACTIONS REPORT

RGD ID: 2520
Species: Rattus norvegicus
RGD Object: Gene
Symbol: Drd2
Name: dopamine receptor D2
Acc ID: CHEBI:2679
Term: amphetamine
Definition: A racemate comprising equimolar amounts of (R)-amphetamine (also known as levamphetamine or levoamphetamine) and (S)-amphetamine (also known as dexamfetamine or dextroamphetamine.
Chemical ID: MESH:D000661
Note: Use of the qualifier "multiple interactions" designates that the annotated interaction is comprised of a complex set of reactions and/or regulatory events, possibly involving additional chemicals and/or gene products.
Object SymbolQualifierEvidenceWithReferenceSourceNotesOriginal Reference(s)
Drd2decreases expressionEXP 6480464CTDAmphetamine results in decreased expression of DRD2 mRNA; Amphetamine results in decreased expression of DRD2 proteinPMID:15183010 PMID:19145071
Drd2increases activityEXP 6480464CTDAmphetamine results in increased activity of DRD2 proteinPMID:7861147
Drd2multiple interactionsEXP 6480464CTDAmphetamine inhibits the reaction [Spiperone binds to DRD2 protein]PMID:2018630
Drd2affects response to substanceISODRD2 (Homo sapiens)6480464CTDDRD2 SNP affects the susceptibility to AmphetaminePMID:19968402
Drd2increases expressionISODrd2 (Mus musculus)6480464CTDAmphetamine results in increased expression of DRD2 mRNA; Amphetamine results in increased expression of DRD2 mRNA alternative formPMID:16916582 PMID:17026527
Drd2increases response to substanceISODrd2 (Mus musculus)6480464CTDDRD2 results in increased susceptibility to AmphetaminePMID:11790512
Drd2multiple interactionsISODrd2 (Mus musculus)6480464CTDCACNA1D protein affects the reaction [Amphetamine results in increased expression of DRD2 mRNA alternative form]PMID:17026527
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