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Term:
tyrosine kinase inhibitor
(CHEBI:38637)
Annotations:
Rat: (11406)
Mouse: (11686)
Human: (12303)
Chinchilla: (0)
Bonobo: (0)
Dog: (2)
Squirrel: (0)
Pig: (11)
Parent Terms
Term With Siblings
Child Terms
protein kinase inhibitor
+
(+)-makassaric acid
(+)-subersic acid
1,4-diamino-2,3-dicyano-1,4-bis(phenylthio)butadiene
1,8-dihydroxy-4-nitroxanthen-9-one
2-(\{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl\}amino)benzamide
aminopurvalanol
Aurora kinase inhibitor
+
CMB4563
CZC8004
DMH1
EC 2.7.10.* (protein-tyrosine kinase) inhibitor
+
EC 2.7.11.* (protein-serine/threonine kinase) inhibitor
+
EC 2.7.11.24 (mitogen-activated protein kinase) inhibitor
+
epidermal growth factor receptor antagonist
+
erlotinib
+
erlotinib hydrochloride
gamma-mangostin
miltefosine
mTOR inhibitor
+
pelitinib
+
piceatannol
+
purvalanol B
quercetin
+
Ro 320-1195
+
salt-inducible kinase 2 inhibitor
+
sangivamycin
tyrosine kinase inhibitor
+
Any protein kinase inhibitor that interferes with the action of tyrosine kinase.
XMD8-92
1-NA-PP1
1-NM-PP1
4,5-dianilinophthalimide
afatinib
+
afatinib dimaleate
axitinib
BE-23372M
biochanin A
+
bosutinib
+
bosutinib hydrate
butein
cabozantinib
+
cabozantinib malate
canertinib
dasatinib (anhydrous)
+
dasatinib monohydrate
DCC-2036
EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor
+
EC 2.7.10.2 (non-specific protein-tyrosine kinase) inhibitor
+
emodin
+
emodin(1-)
genistein
+
herbimycin
hydroxy-2-naphthalenyl-methyl phosphonic acid trisacetoxymethylester
imatinib
+
imatinib methanesulfonate
lapatinib
leflunomide
masitinib
melemeleone B
neratinib
nilotinib
nintedanib
nintedanib esylate
pazopanib
pazopanib hydrochloride
PD173955
+
piceatannol
+
picropodophyllotoxin
ponatinib
PP121
radicicol
regorafenib
+
regorafenib hydrate
SKLB-677
sorafenib
+
teriflunomide
vandetanib
+
WZ4002
Synonyms
Related Synonyms:
TKI inhibitor ; TKI inhibitors ; protein tyrosine kinase inhibitor ; protein tyrosine kinase inhibitors ; tyrosine kinase inhibitors ; tyrphostin ; tyrphostins
Xrefs:
Wikipedia:Tyrosine-kinase_inhibitor