Protein Casr

URN urn:agi-llid:846
Connectivity 336
Name Casr
Description calcium-sensing receptor
Notes The protein encoded by this gene is a G protein-coupled receptor that is expressed in the parathyroid hormone (PTH)-producing chief cells of the parathyroid gland, and the cells lining the kidney tubule. It senses small changes in circulating calcium concentration and couples this information to intracellular signaling pathways that modify PTH secretion or renal cation handling, thus this protein plays an essential role in maintaining mineral ion homeostasis. Mutations in this gene cause familial hypocalciuric hypercalcemia, familial, isolated hypoparathyroidism, and neonatal severe primary hyperparathyroidism. [provided by RefSeq]

Pathway calcium/calcium-mediated signaling pathway
calcium-calcium-mediated signaling pathway
calcium-calcium-mediated signaling pathway
calcium signaling pathway via the calcium-sensing receptor

GO Molecular Function signal transducer activity
phosphoinositide phospholipase C activity
receptor activity
G-protein coupled receptor activity

GO Cellular Component membrane
plasma membrane
integral to membrane
integral to plasma membrane
axon terminus

GO Biological Process positive regulation of cell proliferation
anatomical structure morphogenesis
ossification
vasodilation
signal transduction
calcium-mediated signaling
JNK cascade
positive regulation of ATPase activity
cellular calcium ion homeostasis
chemosensory behavior
detection of calcium ion
regulation of calcium ion transport
calcium ion transport
G-protein coupled receptor protein signaling pathway

Ariadne Ontology GPCR-Gq-iCR

Group GPCR-Gq-iCR
positive regulation of cell proliferation
anatomical structure morphogenesis
ossification
vasodilation
signal transduction
calcium-mediated signaling
JNK cascade
positive regulation of ATPase activity
cellular calcium ion homeostasis
chemosensory behavior
detection of calcium ion
regulation of calcium ion transport
calcium ion transport
G-protein coupled receptor protein signaling pathway
signal transducer activity
phosphoinositide phospholipase C activity
receptor activity
G-protein coupled receptor activity
membrane
plasma membrane
integral to membrane
integral to plasma membrane
axon terminus

MedScan ID 846

Hugo ID 1514

Human chromosome position 3q13

LocusLink ID 846
12374
24247

Alias CAR
FHH
FIH
HHC
EIG8
HHC1
NSHPT
PCAR1
GPRC2A
MGC138441
extracellular calcium-sensing receptor
OTTHUMP00000215576
OTTHUMP00000215577
parathyroid Ca(2+)-sensing receptor 1
parathyroid cell calcium-sensing receptor
cation sensing receptor
G protein coupled receptor, family C, group 2, member A
G protein-coupled receptor, family C, group 2, member A
Calcium-sensing receptor (hypocalciuric hypercalcemia 1 severe neonatal hyperparathyroidism)
Calcium-sensing receptor (hypocalciuric hypercalcemia 1, severe neonatal hyperparathyroidism)
1700108E19Rik
4930562N12
4930562N12Rik
AK039689
calcium sensing receptor, related sequence 4
calcium sensing receptor, related sequence 5
calcium sensing receptor, related sequence IV
calcium sensing receptor, related sequence V
Calcium-sensing receptor
calcium-sensing receptor (hypocalciuric hypercalcemia 1, severe neonatal hy
calcium-sensing receptor related protein 3
calcium-sensing receptor related protein III
Calcium-sensing receptors
CASR
CASR_HUMAN
Casr-rs4
Casr-rs5
cation sensing receptors
Extracellular calcium-sensing receptor precursors
G protein-coupled [Ca(2)](o)-sensing receptor
G protein-coupled [Ca(2+)](o)-sensing receptor
Gprc2a-rs4
Gprc2a-rs5
HHC I
LOC286914
LOC286981
LOC286982
LOC286983
LOC286984
LOC286985
LOC286986
LOC56544
LOC56552
parathyroid Ca(2)-sensing receptor 1
parathyroid Ca(2)-sensing receptor I
parathyroid Ca(2+)-sensing receptor I
parathyroid calcium-sensing receptor 1
parathyroid calcium-sensing receptor I
Parathyroid Cell calcium-sensing receptors
PCAR I
severe neonatal hyperparathyroidism gene

Organism Homo sapiens
Mus musculus
Rattus norvegicus

GenBank ID NC_000003
NM_000388
NP_000379
NT_005612
NW_921807
NW_001838882
NG_009058
AC_000046
AC_000135
NM_001178065
AC068630
AC068754
AY259116
AAP20759
CH471052
EAW79490
EAW79491
EAW79492
DQ088967
AAY68221
DQ327723
ABD04091
DQ327724
ABD04092
DQ327725
ABD04093
DQ327726
ABD04094
DQ327727
ABD04095
DQ327728
ABD04096
S68032
AAB29413
S68033
AAB29414
S68036
AAB29415
X81086
CAA56990
BC104999
AAI05000
BC112236
AAI12237
BP388878
D50855
BAA09453
FJ360896
ACJ04039
S79217
AAB35262
S81755
AAD14370
S83176
AAB46873
U20759
AAA86503
U20760
AAA86504
W56898
P41180
Q2F3K1
Q2F3K2
Q2F3K3
Q2F3K4
Q2F3K5
Q2F3K6
Q86UN7
NC_000082
NM_013803
NP_038831
NT_039624
NW_001030584
AC_000038
AC074229
AF002015
AAC53252
CH466521
EDK97923
EDK97924
AB027140
BAA77688
AF068900
AAC19388
AF092941
AAC62116
AF110178
AAD28371
AF110179
AAD28372
AF128842
AAD40638
AF159565
AAF00193
AK029770
BAC26608
O88982
Q8CDP3
Q9QY96
BC168383
AAI68383
NC_005110
NM_016996
NP_058692
NW_001084662
NW_047356
AC_000079
CH473967
EDM11279
EDM11280
EDM11281
EDM11282
AY214122
AAO59490
U10354
AAC52149
U20289
AAC52195
P48442
Q80ZA8

OMIM ID 601199
612899
239200
146200
145980

Mouse chromosome position 16 26.3 cM

GO ID 0004930
0004435
0004872
0007186
0009653
0019722
0006874
0007635
0005513
0001503
0005887
0005886
0004871
0007254
0006816
0032781
0008284
0051924
0007165
0042311
0043679
0016021
0016020

Rat chromosome position 11q22

Swiss-Prot Accession P41180
Q2F3K1
Q2F3K2
Q2F3K3
Q2F3K4
Q2F3K5
Q2F3K6
Q86UN7
Q8CDP3
Q9QY96
O88982
P48442
Q80ZA8
O08968
O88519
Q9QY95
Q9QZU8
Q9R1D6
Q9R1Y2
Q13912
Q16108
Q16109
Q16110
Q16379
Q2M1T0
Q4PJ19

PIR ID I59362
A56715
B56715

Unigene ID Hs.435615
Mm.103619
Rn.10019

KEGG ID hsa:846
mmu:12374
rno:24247

Swiss-Prot ID CASR_RAT
CASR_MOUSE
CASR_HUMAN
Q8CDP3_MOUSE

Cell Localization Cell membrane
Plasma membrane

IPI ID IPI00190846
IPI00135702
IPI00230189
IPI00012817
IPI00216479
IPI00794666
IPI00569575

Homologene ID 332

RGD ID 2277

MGI ID 1351351