Regulation Adrb1 ---> Heart Failure

URN urn:agi-Regulation:inout-urn:agi-llid:153:out-urn:agi-meshdis:Heart%20Failure::unknown
References 33
Connectivity 2
Effect unknown

TextRef info:pmid/15592928#abs:1
MedLine Reference 15592928:0
Sentence The beta-adrenoceptor (beta-AR) plays an important role in heart failure.

TextRef info:pmid/18425130#abs:1
MedLine Reference 18425130:0
Sentence Beta-adrenergic receptor (betaAR) blockade is a standard therapy for cardiac failure and ischemia.

TextRef info:pmid/9082678#abs:5
MedLine Reference 9082678:4
Sentence Desensitisation of cardiac beta-adrenergic receptors may contribute to contractile dysfunction in chronic heart failure.

TextRef info:pmid/11448139#abs:12
MedLine Reference 11448139:11
Sentence These effects may contribute to beta1-adrenoceptor-mediated cardiotoxicity in heart failure.
CellType cardiomyocyte

TextRef info:pmid/14680448#abs:1
MedLine Reference 14680448:0
Sentence Carvedilol and metoprolol are beta(1)-adrenoceptor antagonists that decrease mortality in heart failure.

TextRef info:pmid/12357106#abs:2
MedLine Reference 12357106:1
Sentence The catecholamines, via alpha- and beta-adrenergic receptor (beta-AR) stimulation, may play a role in the development of heart failure.

TextRef info:pmid/12197595#abs:1
MedLine Reference 12197595:0
Sentence Beta-1-adrenergic receptor (beta1-AR) blockers reduce both the incidence of sudden death and the ventricular volume in heart failure.

TextRef info:pmid/11807612#abs:2
MedLine Reference 11807612:1
Sentence In vitro studies have shown down-regulation of beta-AR density in heart failure and cardiac conditions that may lead to heart failure.

TextRef info:pmid/9456285#abs:8
Organ ventricle
MedLine Reference 9456285:7
Sentence In the right ventricle, beta1-adrenoceptor density decreased only in heart failure; beta2-adrenoceptor density was unchanged.

TextRef info:pmid/19103994#abs:1
MedLine Reference 19103994:0
Sentence Chronic stimulation of the beta(1)-adrenoceptor (beta(1)AR) plays a crucial role in the pathogenesis of heart failure; however, underlying mechanisms remain to be elucidated.

TextRef info:pmid/12954981#abs:2
MedLine Reference 12954981:1
Sentence In addition to regulating cardiac rate and contractility, beta1AR and beta2AR may play different roles in the pathogenesis of heart failure.

TextRef info:pmid/18947427#abs:1
Organ Heart
MedLine Reference 18947427:0
Sentence Persistent stimulation of cardiac beta1-adrenergic receptors by endogenous norepinephrine promotes heart failure progression.

TextRef info:pmid/12422153#abs:1
Organ Heart
MedLine Reference 12422153:0
Sentence Exercise performance in patients with congestive heart failure is partially dependent on cardiac beta1-adrenergic receptor (beta1AR) function.

TextRef info:pmid/10086986#abs:10
Organ Heart
MedLine Reference 10086986:9
Sentence In summary, xamoterol and bucindolol, but not carvedilol and bisoprolol, exhibited direct beta1-adrenoceptor-mediated ISA in normal and heart failure rats.

TextRef info:pmid/11964375#abs:1
MedLine Reference 11964375:0
Sentence Chronic stimulation of the beta(1)-adrenergic receptor leads to hypertrophy and heart failure in beta(1)-adrenergic receptor transgenic mice and contributes to disease progression in heart failure patients.

TextRef info:pmid/18615004#abs:1
MedLine Reference 18615004:0
Sentence Numerous studies have demonstrated that beta(1)- and beta(2)-adrenergic receptor gene (ADRB1 and ADRB2) variants influence cardiovascular risk and beta-blocker responses in hypertension and heart failure.

TextRef info:pmid/12689818#abs:2
Organ Heart
MedLine Reference 12689818:1
Sentence We have, recently, shown that heart-specific overexpression of the beta(1)-adrenergic receptor in transgenic mice (TG) initially leads to increased contractility, followed by LV hypertrophy and heart failure.

TextRef info:pmid/17278500#abs:1
Organ Heart
MedLine Reference 17278500:0
Sentence Myocardial beta adrenergic receptor (beta-AR) concentration can substantially decrease in congestive heart failure and significantly increase in chronic volume overload, such as in severe aortic valve regurgitation.

TextRef info:pmid/16807128#abs:2
Organ Heart
MedLine Reference 16807128:1
Sentence Normalization of betaAR signalling consistently ameliorates cardiac dysfunction and survival in heart failure, suggesting that betaAR dysfunction may be intrinsically linked to the deterioration of cardiac performance.

TextRef info:pmid/17336757#abs:1
Organ Heart
MedLine Reference 17336757:0
Sentence The beta2/beta1 adrenoceptor ratio increases in congestive heart failure (CHF), making the heart relatively more dependent on inotropic, lusitropic, and chronotropic stimulation by the beta2-adrenergic receptor (ADRB2).

TextRef info:pmid/18585502#abs:4
Organ Heart
MedLine Reference 18585502:3
Sentence We analyzed the distribution of autoantibodies against Kv channel-interacting protein (KChIP) 2.6, cardiac troponin I (cTnI), and the beta1-adrenergic receptor (second extracellular loop, cardiac beta1-adrenergic receptor [SEL-beta1-AR])-two other known autoantibodies involved in heart failure.

TextRef info:pmid/15979723#abs:7
Organ Heart
MedLine Reference 15979723:6
Sentence In this review, we attempt to highlight the distinct functionalities and signaling mechanisms of these betaAR subtypes and discuss how these subtype-specific properties of betaARs might affect the pathogenesis of congestive heart failure (CHF) and the therapeutic effectiveness of certain beta-blockers in the treatment of congestive heart failure.

TextRef info:pmid/1323000#abs:2
Organ Heart
MedLine Reference 1323000:1
Sentence With the use of delta Vcfc, a load independent parameter of myocardial contraction, AR mediated contraction was evaluated. beta-AR mediated contraction, delta Vcfc by infusion of a beta-AR agonist, isoproterenol, declined with the advancement of heart failure from 0.41 Circ/sec (NYHA I) to 0.31 (NYHA II), 0.22 (NYHA III) and 0.12 (NYHA IV).

TextRef info:pmid/17158652#cont:201
Organ Heart
MedLine Reference 17158652:10200
Sentence Both apoptosis and ß-AR downregulation are both thought to play a key role in the progression of heart failure.
Journal Heart Circul
Journal Reference v292 i4 p1898
Journal Link http://ajpheart.physiology.org/cgi/content/full/292/4/H1898

TextRef info:pmid/17369456#cont:236
Organ Heart
MedLine Reference 17369456:10235
Sentence Animals with disruption of PI3K? gene are protected from chronic ß-AR stimulation-induced heart failure ( 33 ).
Journal Heart Circul
Journal Reference v293 i1 p385
Journal Link http://ajpheart.physiology.org/cgi/content/full/293/1/H385

TextRef info:pmid/17925438#cont:24
MedLine Reference 17925438:10023
Sentence The ßAR antagonist carvedilol recently was demonstrated to significantly reduce morbidity and mortality in heart failure and in post-AMI patients ( 22 – 25 ).
CellLineName AMI
Journal PNAS
Journal Reference v104 i42 p16657
Journal Link http://www.pnas.org/content/104/42/16657.full

TextRef info:pmid/16699071#cont:22
Organ Nervous system
MedLine Reference 16699071:10021
Sentence Moreover, ß-adrenergic receptor (ß-AR) antagonists have been shown to reduce post-MI remodeling and heart failure development and to improve patients' outcome ( 2 , 19 ).
Journal Heart Circul
Journal Reference v291 i4 p1754
Journal Link http://ajpheart.physiology.org/cgi/content/full/291/4/H1754

TextRef info:pmid/12711600#cont:271
Organ Heart
MedLine Reference 12711600:10270
Sentence These results appear to conflict with observations that betaAR antagonists can reduce fibrosis in heart failure ( 37 , 38 ).
CellType fibroblast
Journal J. Biol. Chem
Journal Reference v278 i27 p24461
Journal Link http://www.jbc.org/cgi/content/full/278/27/24461

TextRef info:pmid/16186489#cont:15
Organ Heart
MedLine Reference 16186489:10014
Sentence Many clinical trials have indicated that angiotensin-converting enzyme inhibitors and ß-AR blockers significantly improve the survival rates of heart failure patients by decreasing cardiac remodeling ( 8 ).
Journal PNAS
Journal Reference v102 i41 p14771
Journal Link http://www.pnas.org/cgi/content/full/102/41/14771

TextRef info:pmid/15569686#cont:262
Organ Heart
MedLine Reference 15569686:10261
Sentence In line with this hypothesis, long term treatment with ß-AR antagonists improves prognosis and cardiac function in heart failure patients ( 47 ), whereas ß-AR agonists increase mortality in these patients ( 48 ).
Tissue Plasma
Journal J. Biol. Chem
Journal Reference v280 i8 p6906
Journal Link http://www.jbc.org/cgi/content/full/280/8/6906

TextRef info:pmid/15001662#cont:225
MedLine Reference 15001662:10224
Sentence The latter authors hypothesized that a 2C - and ß 1 -AR polymorphisms act synergistically to increase synaptic NE release and yield enhanced receptor function, respectively, so as to decrease cardiac function and promote progression of heart failure.
CellLineName GLY
Journal Pharm. Rev
Journal Reference v56 i1 p31
Journal Link http://pharmrev.aspetjournals.org/cgi/content/full/56/1/31

TextRef info:pmid/16204467#cont:131
Organ Heart
MedLine Reference 16204467:10130
Sentence Thus, transgenic overexpression of ß 1 -adrenergic receptors in mice leads to cardiac hypertrophy, heart failure, and early death, whereas, overexpression of the ß 2 -adrenergic receptor actually improves cardiac function and does not adversely affect life span (Xiao et al., 1999b ).
Journal Mol. Pharm
Journal Reference v69 i1 p5
Journal Link http://molpharm.aspetjournals.org/cgi/content/full/69/1/5

TextRef info:pmid/15319203#cont:131
Organ Heart
MedLine Reference 15319203:10130
Sentence The model of increased cavity volumes studied by us is particularly relevant, as it is well recognized that chronic ß-AR activation occurs in chronic heart failure and contributes to increases in cavity volumes and that ß-AR blocking agents reduce cardiac cavity volumes in chronic heart failure ( 5 , 16 ).
Journal Heart Circul
Journal Reference v287 i6 p2762
Journal Link http://ajpheart.physiology.org/cgi/content/full/287/6/H2762