Protein Pik3ca

URN urn:agi-llid:5290
Total Entities 0
Connectivity 1014
Name Pik3ca
Description phosphatidylinositol 3-kinase, catalytic, alpha polypeptide
Notes expression of the human homolog is associated with increased cell proliferation and decreased apoptosis and may play a role in ovarian cancer progression [RGD]

GO Molecular Function 1-phosphatidylinositol-3-kinase activity
phosphatidylinositol 3-kinase activity
1-phosphatidylinositol-4-phosphate 3-kinase activity
phosphatidylinositol-4,5-bisphosphate 3-kinase activity
protein kinase activator activity
transferase activity
transferase activity, transferring phosphorus-containing groups
kinase activity
phosphotransferase activity, alcohol group as acceptor
protein serine-threonine kinase activity
insulin receptor substrate binding
nucleotide binding
ATP binding

GO Cellular Component phosphatidylinositol 3-kinase complex
1-phosphatidylinositol-4-phosphate 3-kinase, class IA complex
intracellular
plasma membrane
cytosol
lamellipodium

GO Biological Process leukocyte migration
Fc-gamma receptor signaling pathway involved in phagocytosis
T cell receptor signaling pathway
innate immune response
Fc-epsilon receptor signaling pathway
T cell costimulation
small molecule metabolic process
phosphatidylinositol biosynthetic process
phosphatidylinositol-3-phosphate biosynthetic process
glucose metabolic process
phospholipid metabolic process
phosphatidylinositol phosphorylation
blood coagulation
platelet activation
cardiac muscle contraction
vasculature development
angiogenesis
endothelial cell migration
regulation of multicellular organism growth
protein kinase B signaling
phosphatidylinositol-mediated signaling
neurotrophin TRK receptor signaling pathway
insulin receptor signaling pathway
fibroblast growth factor receptor signaling pathway
insulin receptor signaling pathway via phosphatidylinositol 3-kinase
epidermal growth factor receptor signaling pathway
negative regulation of fibroblast apoptotic process
negative regulation of neuron apoptotic process
negative regulation of anoikis
positive regulation of protein kinase activity
positive regulation of peptidyl-serine phosphorylation
regulation of genetic imprinting
hypomethylation of CpG island
protein phosphorylation
phosphorylation

Pathway Mechanism of Cetuximab Resistance in Colorectal Cancer
Cowden Syndrome
Mantle Cell Lymphoma Overview
PI3K/AKT/MTOR, NF-kB and BCR Signaling Deregulation in Mantle Cell Lymphoma
Hedgehog Signaling in Mantle Cell Lymphoma
Proteins Involved in Pathogenesis of Breast Cancer Related to ERBB2/VEGFR/Akt Signaling Pathway
Proteins Involved in Pathogenesis of Breast Cancer Related to IGF1R/Akt Signaling Pathway
Breast Cancer Related to IGF1R/Akt Signaling Pathway
Breast Cancer Related to ERBB/VEGFR/Akt Signaling Pathway
Breast Cancer Related to ESR1 Signaling Pathway
Proteins Involved in Pathogenesis of Breast Cancer Related to ESR1 Signaling Pathway
ESR1/ERBB-positive Luminal Breast Cancer
Basal Breast Cancer
Congenital Hypothyroidism Due to Thyroid-Stimulating Hormone Resistance
Thyroid Dysfunction in Graves Disease
Common Non-genomic Effects of Thyroid Hormones
Primary Overt Hypothyroidism Overview
Clear Cell Ovarian Carcinoma
Proteins Involved in Pathogenesis of Clear Cell Ovarian Carcinoma
Mucinous Ovarian Carcinoma
High-grade Serous Ovarian Carcinoma
Proteins Involved in Pathogenesis of Mucinous Ovarian Carcinoma
Proteins Involved in Pathogenesis of High-grade Serous Ovarian Carcinoma
Endometrioid Ovarian Carcinoma
Proteins Involved in Pathogenesis of Endometrioid Ovarian Carcinoma
Ovarian Cancer Overview
Low-grade Serous Ovarian Carcinoma
Proteins Involved in Pathogenesis of Low-grade Serous Ovarian Carcinoma
Type I Endometrial Cancer (Endometrioid Endometrial Cancer)
Type II Endometrial Cancer (Clear-cell Endometrial Cancer and Papillary Serous Endometrial Cancer)
Proteins Involved in Pathogenesis of Endometrial Cancer
Endometrial Cancer Overview
Primary Glioblastoma
Proneural Subtype of Glioblastoma
Growth Factor Signaling in Pancreatic Cancer
Pancreatic Ductal Carcinoma
Pancreatic Neuroendocrine Tumors
Growth Factor Signaling in Hepatocellular Carcinoma
Hepatocellular Carcinoma Overview
Myocardial Remodeling in Myocardial Ischemia
Preconditioning Ischemia
Myocardial Infarction
non-small cell lung cancer pathway
prostate cancer pathway
endometrial cancer pathway
phosphatidylinositol 3-kinase-Akt signaling pathway
phosphatidylinositol 3-kinase-Akt signaling pathway
phosphatidylinositol 3-kinase-Akt signaling pathway

Group PI3K
leukocyte migration
Fc-gamma receptor signaling pathway involved in phagocytosis
T cell receptor signaling pathway
innate immune response
Fc-epsilon receptor signaling pathway
T cell costimulation
small molecule metabolic process
phosphatidylinositol biosynthetic process
phosphatidylinositol-3-phosphate biosynthetic process
1-phosphatidylinositol-3-kinase activity
glucose metabolic process
phospholipid metabolic process
phosphatidylinositol phosphorylation
phosphatidylinositol 3-kinase activity
1-phosphatidylinositol-4-phosphate 3-kinase activity
phosphatidylinositol-4,5-bisphosphate 3-kinase activity
blood coagulation
platelet activation
cardiac muscle contraction
vasculature development
angiogenesis
endothelial cell migration
regulation of multicellular organism growth
protein kinase B signaling
phosphatidylinositol-mediated signaling
neurotrophin TRK receptor signaling pathway
insulin receptor signaling pathway
fibroblast growth factor receptor signaling pathway
insulin receptor signaling pathway via phosphatidylinositol 3-kinase
epidermal growth factor receptor signaling pathway
negative regulation of fibroblast apoptotic process
negative regulation of neuron apoptotic process
negative regulation of anoikis
positive regulation of protein kinase activity
positive regulation of peptidyl-serine phosphorylation
protein kinase activator activity
regulation of genetic imprinting
hypomethylation of CpG island
transferase activity
transferase activity, transferring phosphorus-containing groups
kinase activity
phosphotransferase activity, alcohol group as acceptor
protein serine-threonine kinase activity
protein phosphorylation
phosphorylation
insulin receptor substrate binding
nucleotide binding
ATP binding
phosphatidylinositol 3-kinase complex
1-phosphatidylinositol-4-phosphate 3-kinase, class IA complex
intracellular
plasma membrane
cytosol
lamellipodium
Genes with Mutations Associated with Cowden Syndrome
Genes with Mutations Associated with Mantle Cell Lymphoma
Genes with Mutations Associated with Endometrial Cancer
Genes with Mutations Associated with Hepatocellular Carcinoma
Genes with Mutations, Deletions, and Amplifications Associated with Primary Glioblastoma
Genes with Mutations, Deletions, and Amplifications Associated with Glioma
Biofluids assayable substances

LocusLink ID 5290
18706
170911

Cell Localization Cytoplasm

GO ID 0016303
0035005
0005524
0043560
0016301
0035004
0046934
0030295
0004674
0038095
0038096
0031295
0050852
0001525
0007596
0060048
0043542
0007173
0008543
0006006
0044029
0045087
0008286
0038028
0050900
2000811
0048011
0006661
0046854
0048015
0006644
0030168
0033138
0043491
2000653
0040014
0044281
0001944
0005943
0005829
0030027
0005942
0005886
0000166
0016773
0016740
0016772
2000270
0043524
0036092
0016310
0045860
0006468
0005622
0043066
0006916
0004428
0007165
0005488
0005737
0005739
0005515

Alias MCM
CWS5
MCAP
PI3K
CLOVE
MCMTC
p110-alpha
phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
PI3K-alpha
PI3-kinase p110 subunit alpha
ptdIns-3-kinase subunit p110-alpha
serine/threonine protein kinase PIK3CA
phosphatidylinositol 3-kinase, catalytic, 110-KD, alpha
phosphoinositide-3-kinase, catalytic, alpha polypeptide
phosphatidylinositol 3-kinase, catalytic, alpha polypeptide
phosphatidylinositol-4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, alpha isoform
p110
caPI3K
p110alpha
6330412C24Rik
PI3Kalpha
PI3-kinase subunit alpha
ptdIns-3-kinase subunit alpha
phosphoinositide-3-kinase catalytic alpha polypeptide
phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
PtdIns-3-kinase p110
PIK3CA
PI3K P110-ALPHA
MGC116320
RIKEN cDNA 6330412C24 gene
MGC161268
hydroxykinase
hydroxykinases
MGC142161
MGC142163
OTTMUSP00000023404
6330412C24
Phosphatidylinositol 3-kinase catalytic subunit, alpha isoform
OTTMUSP00000023403

Mouse chromosome position 3 15.7 cM
3 12.4 cM

OMIM ID 171834
612918
615108
162900
114480
114500
114550
182000
211980
602501
603387
167000
613659
137215

Rat chromosome position 2q25

Hugo ID 8975

Human chromosome position 3q26.3

Swiss-Prot Accession P42336
P42337
Q0VGQ5
Q14CW1
Q99762
Q91XL6

PIR ID I38110

GenBank ID NC_000003
NM_006218
NP_006209
NG_012113
NC_018914
AC_000135
ABBA01058543
ABBA01058544
ABBA01058545
ABBA01058546
AC076966
AMYH02008222
CH471052
EAW78423
GM752103
CAV28702
GM865566
CAT16714
AB210020
BAE06102
AK292940
BAF85629
AK297203
BAG59688
AK302608
BAG63856
AU129890
AW445128
BC113601
AAI13602
BC113603
AAI13604
BQ228953
BX437219
BX473473
BX484734
DQ910907
ABI95433
HM437241
ADN43072
U79143
AAB39753
Z29090
CAA82333
P42336
NC_000069
XM_006535409
XP_006535472
XM_006535410
XP_006535473
NM_008839
NP_032865
AC_000025
AAHY01025347
AC110034
AC130281
CH466530
EDL34989
EDL34990
AK018164
AK029399
AK039740
AK051885
AK053528
AK078608
AK151886
AK164801
BC089038
AAH89038
BC130228
AAI30229
U03279
AAA18334
P42337
NC_005101
NM_133399
NP_596890
AC_000070
AABR06015743
AABR06015744
AAHX01016137
AAHX01016138
AF395897
AAK83379
BC086516
BC099154
BP500486
BQ203660
CB793501
CK366194
CK366305
CR754046
DV722574
DV728106
DY314099
FM035395
FM096453
XM_001063573
XP_001063573
NW_047625
NW_001084800
XM_001059350
XP_001059350
Q91XL6
XM_001059407
XP_001059407
XM_001059296
XP_001059296
AAH99154
Q4KLK3

Unigene ID Hs.553498
Hs.715194
Mm.260521
Rn.44193
Rn.190480
Rn.165275

KEGG ID hsa:5290
mmu:18706
rno:170911

Swiss-Prot ID PK3CA_MOUSE
PK3CA_HUMAN

EC Number 2.7.1.153
2.7.11.1
2.7.1.137

Ensembl ID ENSMUSG00000027665
ENSMUSP00000029201
ENSMUST00000029201
ENSMUSP00000103878
ENSMUST00000108243
ENSRNOG00000010458
ENSRNOP00000014527
ENSRNOT00000014527

Homologene ID 21249

Organism Homo sapiens
Mus musculus
Rattus norvegicus

MGI ID 1206581

RGD ID 620916

MedScan ID 5290
170911

Primary Cell Localization Cytoplasm

IPI ID IPI00309224
IPI00031386
IPI00781719
IPI00779888
IPI00211380
IPI00769166
IPI00769069
IPI00766767