Protein Pik3ca

URN urn:agi-llid:5290
Total Entities 0
Connectivity 538
Name Pik3ca
Description phosphatidylinositol 3-kinase, catalytic, alpha polypeptide
Notes expression of the human homolog is associated with increased cell proliferation and decreased apoptosis and may play a role in ovarian cancer progression [RGD]

Ariadne Ontology PI3K
Secreted proteins

GO Molecular Function insulin receptor substrate binding
nucleotide binding
ATP binding
transferase activity
transferase activity, transferring phosphorus-containing groups
phosphotransferase activity, alcohol group as acceptor
kinase activity
1-phosphatidylinositol-3-kinase activity
protein serine-threonine kinase activity
protein kinase activator activity
phosphatidylinositol-4,5-bisphosphate 3-kinase activity
phosphatidylinositol 3-kinase activity

GO Cellular Component phosphatidylinositol 3-kinase complex
1-phosphatidylinositol-4-phosphate 3-kinase, class IA complex
cytosol
lamellipodium

GO Biological Process protein kinase B signaling cascade
phosphatidylinositol-mediated signaling
T cell receptor signaling pathway
nerve growth factor receptor signaling pathway
fibroblast growth factor receptor signaling pathway
insulin receptor signaling pathway
epidermal growth factor receptor signaling pathway
insulin receptor signaling pathway via phosphatidylinositol 3-kinase cascade
positive regulation of peptidyl-serine phosphorylation
positive regulation of protein kinase activity
regulation of genetic imprinting
hypomethylation of CpG island
negative regulation of apoptotic process
negative regulation of anoikis
T cell costimulation
platelet activation
protein phosphorylation
phospholipid metabolic process
phosphatidylinositol phosphorylation
phosphatidylinositol biosynthetic process
phosphorylation
endothelial cell migration
leukocyte migration
regulation of multicellular organism growth
angiogenesis
vasculature development
cardiac muscle contraction
blood coagulation
glucose metabolic process
small molecule metabolic process

Pathway non-small cell lung cancer pathway
phosphatidylinositol 3-kinase-Akt signaling pathway
endometrial cancer pathway
prostate cancer pathway
endometrial cancer pathway
phosphatidylinositol 3-kinase-Akt signaling pathway
non-small cell lung cancer pathway
prostate cancer pathway

Group PI3K
protein kinase B signaling cascade
phosphatidylinositol-mediated signaling
T cell receptor signaling pathway
nerve growth factor receptor signaling pathway
fibroblast growth factor receptor signaling pathway
insulin receptor signaling pathway
epidermal growth factor receptor signaling pathway
insulin receptor signaling pathway via phosphatidylinositol 3-kinase cascade
positive regulation of peptidyl-serine phosphorylation
positive regulation of protein kinase activity
regulation of genetic imprinting
hypomethylation of CpG island
negative regulation of apoptotic process
negative regulation of anoikis
T cell costimulation
platelet activation
protein phosphorylation
phospholipid metabolic process
phosphatidylinositol phosphorylation
phosphatidylinositol biosynthetic process
phosphorylation
endothelial cell migration
leukocyte migration
regulation of multicellular organism growth
angiogenesis
vasculature development
cardiac muscle contraction
blood coagulation
glucose metabolic process
small molecule metabolic process
insulin receptor substrate binding
nucleotide binding
ATP binding
transferase activity
transferase activity, transferring phosphorus-containing groups
phosphotransferase activity, alcohol group as acceptor
kinase activity
1-phosphatidylinositol-3-kinase activity
protein serine-threonine kinase activity
protein kinase activator activity
phosphatidylinositol-4,5-bisphosphate 3-kinase activity
phosphatidylinositol 3-kinase activity
phosphatidylinositol 3-kinase complex
1-phosphatidylinositol-4-phosphate 3-kinase, class IA complex
cytosol
lamellipodium
Secreted proteins

MedScan ID 5290
170911

Hugo ID 8975

Human chromosome position 3q26.3

GenBank ID NC_000003
NM_006218
NP_006209
NG_012113
NC_018914
AC_000135
AC076966
CH471052
EAW78423
GM752103
CAV28702
GM865566
CAT16714
AB210020
BAE06102
AK292940
BAF85629
AK297203
BAG59688
AK302608
BAG63856
AU129890
AW445128
BC113601
AAI13602
BC113603
AAI13604
BQ228953
BX437219
BX473473
BX484734
DQ910907
ABI95433
HM437241
ADN43072
U79143
AAB39753
Z29090
CAA82333
P42336
NC_000069
NM_008839
NP_032865
AC_000025
AC110034
AC130281
CH466530
EDL34989
EDL34990
AK018164
AK029399
AK039740
AK051885
AK053528
AK078608
AK151886
AK164801
BC089038
AAH89038
BC130228
AAI30229
U03279
AAA18334
P42337
NC_005101
NM_133399
NP_596890
AC_000070
AF395897
AAK83379
BC086516
BC099154
BP500486
BQ203660
CB793501
CK366194
CK366305
CR754046
DV722574
DV728106
DY314099
FM035395
FM096453
XM_001063573
XP_001063573
NW_047625
NW_001084800
XM_001059350
XP_001059350
Q91XL6
XM_001059407
XP_001059407
XM_001059296
XP_001059296
AAH99154
Q4KLK3

LocusLink ID 5290
18706
170911

Alias PI3K
CLOVE
p110-alpha
phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
PI3K-alpha
PI3-kinase p110 subunit alpha
ptdIns-3-kinase subunit p110-alpha
serine/threonine protein kinase PIK3CA
phosphatidylinositol 3-kinase, catalytic, 110-KD, alpha
phosphoinositide-3-kinase, catalytic, alpha polypeptide
phosphatidylinositol 3-kinase, catalytic, alpha polypeptide
phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha
phosphatidylinositol-4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, alpha isoform
p110
caPI3K
p110alpha
6330412C24Rik
PI3Kalpha
PI3-kinase subunit alpha
ptdIns-3-kinase subunit alpha
phosphoinositide-3-kinase catalytic alpha polypeptide
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
PI3K P110-ALPHA
PIK3CA
PtdIns-3-kinase p110
hydroxykinases
Phosphatidylinositol 3-kinase catalytic subunit, alpha isoform
hydroxykinase
6330412C24
MGC142161
MGC142163
MGC161268
OTTMUSP00000023403
OTTMUSP00000023404
MGC116320

Organism Homo sapiens
Mus musculus
Rattus norvegicus

OMIM ID 171834
612918
162900
114480
114500
137215
182000
114550
211980
167000

Unigene ID Hs.553498
Hs.715194
Mm.260521
Rn.44193
Rn.190480
Rn.165275

KEGG ID hsa:5290
mmu:18706
rno:170911

Swiss-Prot Accession P42336
P42337
Q0VGQ5
Q14CW1
Q99762
Q91XL6

EC Number 2.7.1.153
2.7.11.1
2.7.1.137

GO ID 0016303
0005524
0043560
0016301
0035004
0046934
0030295
0004674
0031295
0050852
0001525
0007596
0060048
0043542
0007173
0008543
0006006
0044029
0008286
0038028
0050900
2000811
0048011
0006661
0046854
0048015
0006644
0030168
0033138
0043491
2000653
0040014
0044281
0001944
0005943
0005829
0030027
0005942
0000166
0016773
0016740
0016772
0043066
0016310
0006468
0006916
0045860
0004428
0007165
0005488
0005737
0005739
0005515

PIR ID I38110

Swiss-Prot ID PK3CA_MOUSE
PK3CA_HUMAN

Cell Localization Cytoplasm

IPI ID IPI00309224
IPI00031386
IPI00781719
IPI00779888
IPI00211380
IPI00769166
IPI00769069
IPI00766767

Mouse chromosome position 3 12.4 cM

Rat chromosome position 2q25

Homologene ID 21249

MGI ID 1206581

RGD ID 620916

Primary Cell Localization Cytoplasm