Protein Crebbp

URN urn:agi-llid:1387
Connectivity 563
Name Crebbp
Description CREB binding protein
Notes A missense mutation has been identified in codon 1175 of CREBBP in a mild case of Rubinstein-Taybi syndrome. A missense mutation has been identified in codon 1175 of CREBBP in a mild case of Rubinstein-Taybi syndrome. CBP acetylation controls HNF6 protein stability. CBP and p300 function as co-activators of Sox9 for cartilage tissue-specific gene expression and chondrocyte differentiation. CBP enhances tumor necrosis alpha-induced cell death in rheumatoid synoviocytes. CBP has a role in regulating 5-aminolevulinate synthase gene expression via the AP-1 complex in human tumor cells. CBP-induced acetylation of AFX is a novel modification mechanism by which AFX keeps the transcriptional activity mitigating in the nucleus. Direct involvement of CREB-binding protein/p300 in sequence-specific DNA binding of virus-activated interferon regulatory factor-3 holocomplex. E2A-PBX1 interacts directly with the KIX domain of CBP/p300 in the induction of proliferation in primary hematopoietic cells. Estrogen receptor-alpha represses human GnRH receptor gene transcription via an indirect mechanism involving Creb-binding protein. GCMa acetylation is mediated by CBP, which stimulates GCMa transcriptional activity through cyclic AMP/protein kinase A signaling. HIF-1alpha, STAT3, CBP/p300 and Ref-1/APE regulate Src-dependent hypoxia-induced expression of VEGF in pancreatic and prostate carcinomas. HIV Tat is a general inhibitor of histone acetylation by cellular HATs and for the CREB-binding protein (CBP), it induces a substrate selectivity. IL-6-inducible expression of the hAGT promoter is mediated by physical association of the COOH terminus of STAT3 with p300/CBP, the recruitment of which targets histone acetylation and results in chromatin remodeling. In 92 patients, we were able to identify a total of 36 mutations in CBP. By using multiple ligation-dependent probe amplification, we found not only several deletions but also the first reported intragenic duplication in a patient with RSTS. In conclusion, this research supports FSCN1 as a novel marker of NT2 neuronal differentiation and the possible role of CBP in its regulation. Interaction of PIMT with transcriptional coactivators CBP, p300, and PBP differential role in transcriptional regulation. Loss of CREBBP was not statistically significant selection in cancer cells stratified by various criteria for the concordant loss of EP300 and CREBBP. Loss of heterozygosity and internal tandem duplication mutations of the CBP gene are frequent events in human esophageal squamous cell carcinoma. Mutations and deletions of the CBP gene is associated with lung cancer. Novel heterozygous deletion in CREBBP in Rubinstein-Taybi syndrome patient results in the loss of exon 30. Oct-1 potentiates CREB-dependent cyclin D1 transcriptional activity by a phospho-CREB and CREB binding protein-independent mechanism. PHD finger mutations cause a loss of CBP acetyltransferase activity. Recruitment of Daxx following SUMO modification represents a previously undescribed mechanism in modulating CREB-binding protein (CBP) transcriptional potential. Regulatory motifs for CREB-binding protein and Nfe2l2 transcription factors in the upstream enhancer of the mitochondrial uncoupling protein 1 gene. Smad-binding peptide aptamers can be developed to selectively inhibit TGF-beta-induced gene expression. Smad3 induces chondrogenesis through the activation of SOX9 via CREB-binding protein/p300 recruitment. Suppression of CBP in human mammary epithelial cells results in loss of reconstituted extracellular matrix-mediated growth control and apoptosis and loss of laminin-5 alpha 3-chain expression. The CBP/p300 acetylase and the CARM1 methyltransferase can positively regulate the expression of estrogen-responsive genes, there is a crosstalk between lysine acetylation and arginine methylation on chromatin. The KID-interacting domain of human coactivator CREB-binding protein (CBP) is the CBP domain that is targeted by HIV-1 Tat during HIV-1 propagation. The PHD type zinc finger is an integral part of the CBP acetyltransferase domain. The fact that Egr-1 promoter/reporter gene transcription is upregulated by a constitutively active CREB mutant indicates that the CRE couples other signaling cascades via CREB to the Egr-1 gene. The interaction between CtBP and CBP is functionally important and leads to impairment of histone H3 acetylation by CBP at specific lysine residues (Lys9, Lys14, and Lys18) in a dose-dependent and NADH-dependent manner. The interaction of fibroblast growth factor receptor-1: wiwth CREb binding protein allows activation of gene transcription and may play a role in cell differentiation. The site of the KID-interacting (KIX) domain of CBP that recognizes c-Jun and mixed lineage leukemia MLL proteins is identified as the same site that binds HIV-1 Tat protein. We aimed to determine the rate of point mutations and other small molecular lesions in true Rubinstein-Taybi syndrome and possible mild variants, by using genomic DNA sequencing of the CREBBP gene. Activation of CREB-binding protein and inhibition of MAPK has a role in cAMP-dependent protein kinase type I regulation of ethanol-induced cAMP response element-mediated gene expression. Activity of ESE-1 is positively and negatively modulated by other interacting proteins including Ku70, Ku86, p300, and CBP. Arginine methylation of CBP is required for IFN-gamma induction of MHC-II. A kinetic analysis shows that CIITA, CARM1, and H3-R17 methylation all precede CBP loading on the MHC-II promoter during IFN-gamma treatment. Arginine methylation represents an important mechanism for modulating CBP co-activator transcriptional activity. Deletion of the CBP bromo- and C/H3 domains eliminates stimulation of nucleosomal histone deacetylase activity in vitro and transcriptional coactivation by EBV Zta in transfected cells. Effect of CREB-binding protein on inhibition of Smad-mediated transcriptional activation by K-bZIP was examined. Glutamine rich and bZIP domains stabilize CREB binding to chromatin. Important functions in coordinated cell cycle progression. In human mammary epithelial cells, CBP/p300 were both modulated by an all-trans-retinoic acid (ATRA) signaling pathway and were required for a normal response to ATRA. Interaction of CREB-binding protein with EWS selectively activates hepatocyte nuclear factor 4-mediated transcription. Is co-expressed with CREB and CBP in extravillous cytotrophoblasts, revealing the in vivo relevance of this transactivation pathway. Overexpression of CBP is detected from the very early stages of laryngeal carcinogenesis, suggesting that CBP may play a role in malignant transformation of precancerous laryngeal lesions. P34SEI-1 strongly suppressed CREB-mediated transcription, and this suppression was overcome by excess amount of CBP. Recruitment to pp90RSK regulates cAMP response element-binding protein activity which is negatively affected by ERK phosphorylation. Results suggest that all-trans-retinoic acid and retinoic acid receptors regulate growth arrest of human mammary epithelial cells and modulate CBP/p300 protein expression. Role in acetylation of beta-catenin. Role in transcriptional control of the inflammatory response. Structurally distinct modes of recognition of the KIX domain of this protein by Jun and CREB. Substrate specificity; structure activity relationship. The conserved bromo-domain of the transcriptional coactivator CBP (CREB binding protein) binds specifically to p53 at the C-terminal acetylated lysine 382. The histone chaperone SET regulates CBP-mediated transcription.

Pathway FGFR -> AP-1/CREB/CREBBP/ELK-SRF/MYC signaling
T-cell receptor -> CREBBP signaling
canonical Wnt signaling pathway
altered canonical Wnt signaling pathway
canonical Wnt signaling pathway
altered canonical Wnt signaling pathway
hypoxia inducible factor pathway

GO Molecular Function signal transducer activity
chromatin binding
transferase activity
transcription activator activity
transcription factor activity
transcription cofactor activity
transcription factor binding
p53 binding
SMAD binding
DNA binding
peroxisome proliferator activated receptor binding
transcription coactivator activity
MyoD binding
metal ion binding
zinc ion binding
acetyltransferase activity
histone acetyltransferase activity

GO Cellular Component protein complex
cytoplasm
outer kinetochore of condensed chromosome
nuclear body
transcription factor complex
histone acetyltransferase complex
PML body
nucleus

GO Biological Process cell proliferation
interspecies interaction between organisms
germ-line stem cell maintenance
signal transduction
regulation of S phase
regulation of transcription
positive regulation of transcription
positive regulation of transcription, DNA-dependent
positive regulation of transcription from RNA polymerase II promoter
regulation of transcription, DNA-dependent
positive regulation of transcription factor activity
transcription
histone acetylation
N-terminal peptidyl-lysine acetylation
response to hypoxia
protein complex assembly
homeostatic process

Ariadne Ontology Transcription factors

Group Transcription factors
cell proliferation
interspecies interaction between organisms
germ-line stem cell maintenance
signal transduction
regulation of S phase
regulation of transcription
positive regulation of transcription
positive regulation of transcription, DNA-dependent
positive regulation of transcription from RNA polymerase II promoter
regulation of transcription, DNA-dependent
positive regulation of transcription factor activity
transcription
histone acetylation
N-terminal peptidyl-lysine acetylation
response to hypoxia
protein complex assembly
homeostatic process
signal transducer activity
chromatin binding
transferase activity
transcription activator activity
transcription factor activity
transcription cofactor activity
transcription factor binding
p53 binding
SMAD binding
DNA binding
peroxisome proliferator activated receptor binding
transcription coactivator activity
MyoD binding
metal ion binding
zinc ion binding
acetyltransferase activity
histone acetyltransferase activity
protein complex
cytoplasm
outer kinetochore of condensed chromosome
nuclear body
transcription factor complex
histone acetyltransferase complex
PML body
nucleus

MedScan ID 1387

Hugo ID 2348

Human chromosome position 16p13.3

LocusLink ID 1387
12914
54244
436331

Alias CBP
RSTS
KAT3A
CREB-binding protein
AW558298
CBP/p300
p300/CBP
RTS
cAMP response element binding protein binding protein
cAMP response element-binding protein binding protein
cAMP response element-binding protein-binding protein
cAMP responsive element binding protein binding protein
cAMP responsive element-binding protein binding protein
cAMP responsive element-binding protein-binding protein
cAMP-response element binding protein binding protein
cAMP-response element-binding protein binding protein
cAMP-response element-binding protein-binding protein
CBP_MOUSE
CREB binding protein
CREBBP
cyclic AMP response element binding protein binding protein
cyclic AMP response element-binding protein binding protein
cyclic AMP response element-binding protein-binding protein
cyclic AMP responsive element binding protein binding protein
cyclic AMP responsive element-binding protein binding protein
cyclic AMP responsive element-binding protein-binding protein
cyclic AMP-response element binding protein binding protein
cyclic AMP-response element-binding protein binding protein
cyclic AMP-response element-binding protein-binding protein
histone acetyltransferase CBP
LOC436331
LOC497663
LOC547230
Rubinstein-Taybi syndrome gene
Rubinstein-Taybi syndrome protein
Creb binding protein (CBP)
similar to CREB-binding protein

Organism Homo sapiens
Mus musculus
Rattus norvegicus

GenBank ID NC_000016
NM_001079846
NP_001073315
NM_004380
NP_004371
NT_010393
NW_926018
NW_001838341
NG_009873
AC_000059
AC_000148
AC004509
AAC08447
AC004651
AC004760
AAC17736
AC006111
AC007151
CH471112
EAW85334
EAW85335
EAW85336
EAW85337
CS330044
CAL00150
AB210043
BAE06125
AK124320
AK304771
BAG65526
BC036486
AAH36486
U47741
AAC51770
U85962
AAC51331
U89354
AAC51339
U89355
AAC51340
O60424
Q4G0V0
Q4LE28
Q712H6
Q75MY6
Q92793
NC_000082
NM_001025432
NP_001020603
NT_039624
NW_001030584
AC_000038
AC132380
AY079443
AAL87531
AY079444
AAL87532
CAAA01026247
CH466521
EDK97225
AK048818
BAE20666
AK051071
AK136057
AK162593
BC010297
BC072594
AAH72594
BU705617
S66385
AAB28651
P45481
Q3V351
Q6GQV9
Q8QZV8
BC172737
AAI72737
NC_005109
NM_133381
NP_596872
NW_047333
NW_001084654
AC_000078
AF410812
AAN39140
AF410813
AAN39141
AB066219
BAB62424
AY462245
AAR23149
Q6JHU9
Q812C1
Q812C2
Q91XT1
NT_037887
BG074283
AW558298
BG069466
AI507501
BG080014
NW_000107
BG076163
AI431079

OMIM ID 600140
180849

Mouse chromosome position 16 A1

GO ID 0051577
0046332
0016407
0003682
0004402
0046872
0002039
0042975
0004871
0003713
0003700
0008134
0016740
0008270
0018076
0008283
0030718
0016573
0042592
0044419
0045941
0045944
0006461
0033261
0045449
0006355
0001666
0007165
0005737
0000123
0016604
0005634
0000940
0005667
0003677
0016563
0003712
0051091
0045893
0006350
0016605
0043234
0005515

Rat chromosome position 10q12

Swiss-Prot Accession Q4LE28
Q92793
O60424
Q4G0V0
Q712H6
Q75MY6
Q6GQV9
P45481
Q3V351
Q8QZV8
Q6JHU9
Q812C1
Q812C2
Q91XT1
O00147
Q16376
D3DUC9

PIR ID S39162

Unigene ID Hs.459759
Mm.132238
Mm.392384
Rn.12815
Rn.108128
Mm.387139
Mm.392739
Mm.386759
Mm.393135

KEGG ID hsa:1387
mmu:12914
rno:54244

EC Number 2.3.1.48

Swiss-Prot ID CBP_HUMAN
Q4LE28_HUMAN
D3DUC9_HUMAN
Q6GQV9_MOUSE
Q6JHU9_RAT

Cell Localization Nucleus

IPI ID IPI00023339
IPI00619932
IPI00463549
IPI00155855
IPI00875480
IPI00652158
IPI00751842
IPI00421436
IPI00781902

Homologene ID 68393

RGD ID 2401

MGI ID 1098280