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GENE - CHEMICAL INTERACTIONS REPORT

RGD ID: 2803
Species: Rattus norvegicus
RGD Object: Gene
Symbol: Hmgcr
Name: 3-hydroxy-3-methylglutaryl-CoA reductase
Acc ID: CHEBI:41774
Term: tamoxifen
Definition: A stilbenoid that has formula 371.51460.
Chemical ID: MESH:D013629
Note: Use of the qualifier "multiple interactions" designates that the annotated interaction is comprised of a complex set of reactions and/or regulatory events, possibly involving additional chemicals and/or gene products.
Object SymbolQualifierEvidenceWithReferenceSourceNotesOriginal Reference(s)
Hmgcraffects expressionISOHmgcr (Mus musculus)6480464CTDTamoxifen affects the expression of HMGCR mRNAPMID:20937368
Hmgcrincreases expressionISOHmgcr (Mus musculus)6480464CTDTamoxifen results in increased expression of HMGCR mRNA; Tamoxifen results in increased expression of HMGCR proteinPMID:35944649
Hmgcrmultiple interactionsISOHmgcr (Mus musculus)6480464CTDfatostatin inhibits the reaction [Tamoxifen results in increased expression of HMGCR mRNA]; fatostatin inhibits the reaction [Tamoxifen results in increased expression of HMGCR protein]PMID:35944649
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